Template:Affinities of selected androgen receptor ligands

v
t
e
Affinities^[a]^[1]
Compound	RBATooltip Relative binding affinity^[b]
Metribolone	100
Dihydrotestosterone	85
Cyproterone acetate	7.8
Bicalutamide	1.4
Nilutamide	0.9
Hydroxyflutamide	0.57
Flutamide	<0.0057
Notes: ↑ At androgen receptors; measured in human prostate tissue. ↑ Relative to Metribolone, which is by definition 100%

References

↑ Ayub M, Levell MJ (August 1989). "The effect of ketoconazole related imidazole drugs and antiandrogens on [3H] R 1881 binding to the prostatic androgen receptor and [3H]5 alpha-dihydrotestosterone and [3H]cortisol binding to plasma proteins". J. Steroid Biochem. 33 (2): 251–5. doi:10.1016/0022-4731(89)90301-4. PMID 2788775.